APINAC

APINAC
Clinical data
Other namesAKB-57, AKB57
Legal status
Legal status
Identifiers
  • N-(1-Adamantyl)-1-pentylindazole-3-carboxylate
CAS Number
PubChem CID
ChemSpider
UNII
CompTox Dashboard (EPA)
Chemical and physical data
FormulaC23H31N2O2
Molar mass367.513 g·mol−1
3D model (JSmol)
  • CCCCCn1nc(C(=O)OC23CC4CC(CC(C4)C2)C3)c2ccccc21
  • InChI=1S/C23H30N2O2/c1-2-3-6-9-25-20-8-5-4-7-19(20)21(24-25)22(26)27-23-13-16-10-17(14-23)12-18(11-16)15-23/h4-5,7-8,16-18H,2-3,6,9-15H2,1H3
  • Key:KCCVWUAAHDXNNQ-UHFFFAOYSA-N

APINAC (AKB-57, N-(1-adamantyl)-1-pentylindazole-3-carboxylate) is a drug that acts as an agonist for the cannabinoid receptors.[2] It was detected in Slovenia in 2016[3] and is on the UNODC list of synthetic cannabinoids.[4]

Legality

APINAC is covered by the UK blanket ban on synthetic cannabinoids.

Detection

APINAC can be bought by labs as a reference standard.[5] APINAC metabolizes to N-pentylindazole-3-carboxylic acid, hydroxylated N-pentylindrazole-3-carboxylic acid, and 1-adamantanol in rats.[2]

See also

References

  1. ^ Anvisa (2023-07-24). "RDC Nº 804 - Listas de Substâncias Entorpecentes, Psicotrópicas, Precursoras e Outras sob Controle Especial" [Collegiate Board Resolution No. 804 - Lists of Narcotic, Psychotropic, Precursor, and Other Substances under Special Control] (in Brazilian Portuguese). Diário Oficial da União (published 2023-07-25). Archived from the original on 2023-08-27. Retrieved 2023-08-27.
  2. ^ a b Savchuk S, Appolonova S, Pechnikov A, Rizvanova L, Shestakova K, Tagliaro F (2017-07-01). "In vivo metabolism of the new synthetic cannabinoid APINAC in rats by GC–MS and LC–QTOF-MS". Forensic Toxicology. 35 (2): 359–368. doi:10.1007/s11419-017-0364-y. ISSN 1860-8973.
  3. ^ "Analytical Report, AKB-57 (C23H30N2O2)" (PDF). NPS AND RELATED COMPOUNDS DATABASE. Slovenian National Forensic Laboratory (NFL) (published 2016-02-12). 2016-02-04. adamantan-1-yl 1-pentyl-1H-indazole-3-carboxylate; KCCVWUAAHDXNNQ-UHFFFAOYSA-N
  4. ^ "Substance Details AKB-57". www.unodc.org. Retrieved 2026-06-26.
  5. ^ "Apinac (CAS 2219331-93-6)". Cayman. Retrieved 2026-06-26.

Content Disclaimer

Informasi ini disarikan dari Wikipedia dan disajikan kembali untuk tujuan edukasi. Konten tersedia di bawah lisensi CC BY-SA 3.0. Kami tidak bertanggung jawab atas ketidakakuratan data yang bersumber dari kontribusi publik tersebut.

  1. The information displayed on this website is sourced in part or in whole from Wikipedia and has been adapted for the purpose of restating it. We strive to provide accurate and relevant information, however:
  2. There is no guarantee of absolute accuracy. Wikipedia is an open, collaborative project that can be edited by anyone, so information is subject to change.
  3. It is not intended to constitute professional advice. The content displayed is for informational and educational purposes only. For important decisions (e.g., medical, legal, or financial), please consult a professional.
  4. Content copyright. Wikipedia is licensed under the Creative Commons Attribution-ShareAlike License (CC BY-SA). This means that content may be reused with appropriate attribution and shared under a similar license.
  5. Responsible use. Any risk arising from the use of information from this website is entirely the responsibility of the user.